Improved Synthetic Route to Methyl 1-Fluoroindan-1-carboxylate (FICA Me Ester) and 4-Methyl Derivatives
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چکیده
منابع مشابه
A simple synthetic route to methyl 3-fluoropyridine-4-carboxylate by nucleophilic aromatic substitution.
The nitro group of methyl 3-nitropyridine-4-carboxylate (1) has successfully been replaced by fluoride anion via nucleophilic aromatic substitution to give the 3-fluoro- pyridine-4-carboxylate 2.
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ژورنال
عنوان ژورنال: Chemical and Pharmaceutical Bulletin
سال: 2014
ISSN: 0009-2363,1347-5223
DOI: 10.1248/cpb.c14-00192